- |||||||||| Journal: Potential mechanisms and drug prediction of Rheumatoid Arthritis and primary Sj (Pubmed Central) - Feb 19, 2024
In conclusion, we identified commom targets as potential biomarkers in RA and pSS from publicly available databases and predicted potential drugs based on the targets. A new understanding of the molecular mechanisms associated with RA and pSS is provided according to the miRNA-gene network.
- |||||||||| Tepezza (teprotumumab) / Roche, Amgen
Journal: Objective Diplopia Outcomes for Patients Treated With Teprotumumab for Thyroid Eye Disease. (Pubmed Central) - Feb 19, 2024 There are some baseline measures, such as CAS and right and left gaze horizontal prism deviation that can help better predict how a patient will respond to teprotumumab treatment. Our results can better inform physicians of how to counsel patients with TED when considering teprotumumab therapy.
- |||||||||| Krazati (adagrasib) / BMS, Lumakras (sotorasib) / Amgen
Review, Journal: Multiple medicinal chemistry strategies of targeting KRAS: State-of-the art and future directions. (Pubmed Central) - Feb 19, 2024 We systematically summarize recent advances in the discovery and optimization processes of direct KRAS inhibitors (including KRAS, KRAS, KRAS and KRAS inhibitors), indirect KRAS inhibitors (SOS1 and SHP2 inhibitors), pan-KRAS inhibitors, as well as proteolysis-targetingchimeras degrades and molecular chaperone modulators from the perspective of medicinal chemistry. We also discuss the current challenges and opportunities of KRAS inhibition and hope to shed light on future KRAS drug discovery.
- |||||||||| ivabradine / Generic mfg.
Journal: Ivabradine for congenital ectopic tachycardia in newborn. (Pubmed Central) - Feb 19, 2024 Congenital junctional ectopic tachycardia is rare, and it is mostly resistant to the conventional treatment.Ivabradine is a new anti-arrhythmic agent, used extensively to decrease sinus rate in the treatment of cardiac failure. Ivabradine may be an option for the resistant congenital ectopic tachycardia.
- |||||||||| Ibrance (palbociclib) / Pfizer, giredestrant (GDC-9545) / Roche
Journal, Metastases: Phase Ia/b Study of Giredestrant (Pubmed Central) - Feb 19, 2024 P1 Giredestrant was well tolerated and clinically active in patients who progressed on prior ET. Results warrant further evaluation of giredestrant in randomized trials in early- and late-stage ER+ breast cancer.
- |||||||||| Jakafi (ruxolitinib) / Incyte, Neupogen (filgrastim) / Kyowa Kirin, Amgen
Trial completion date, Trial primary completion date, Metastases: Reduced Intensity Allogeneic HCT in Advanced Hematologic Malignancies w/T-Cell Depleted Graft (clinicaltrials.gov) - Feb 19, 2024 P1, N=40, Recruiting, Trial completion date: Sep 2024 --> Dec 2024 | Trial primary completion date: Jun 2024 --> Dec 2024 Trial completion date: Jun 2024 --> Dec 2025 | Trial primary completion date: Jun 2024 --> Dec 2025
- |||||||||| Truxima (rituximab-abbs) / Indukern, Teva, Mundipharma, Celltrion, Nippon Kayaku, Neupogen (filgrastim) / Kyowa Kirin, Amgen, Rituxan (rituximab) / Roche
Trial completion date: NCI-2011-00344: Genetically Engineered Lymphocyte Therapy After Peripheral Blood Stem Cell Transplant in Treating Patients With High-Risk, Intermediate-Grade, B-cell Non-Hodgkin Lymphoma (clinicaltrials.gov) - Feb 18, 2024 P1/2, N=8, Active, not recruiting, Trial completion date: Jun 2024 --> Dec 2025 | Trial primary completion date: Jun 2024 --> Dec 2025 Trial completion date: Dec 2023 --> Dec 2024
- |||||||||| Prolia (denosumab) / Amgen
Giant Cell Tumor of Bone with H3F3A Mutation and Unusual Bone Formation; Features to Separate from Low-Grade Central Osteosarcoma (Exhibit Hall; Poster Board Number: 80) - Feb 18, 2024 - Abstract #USCAP2024USCAP_1193; GCT-UBF generally exhibits separate fragments of non-lacelike woven bone, mild to moderate cellularity, rare to absent osteoclast-type giant cells or mitoses, H3F3A mutation and flat copy number changes, with lack of significant atypia, necrosis, additional pathogenic gene alterations or MDM2 amplification, distinguishing these from LG-OSA. A small subset with atypical features and multiple copy number alterations raise concern for malignancy and require further study.
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen
To B or Not to B: Utility of PAX5 in Lineage Assignment of Acute Leukemia (Exhibit Hall; Poster Board Number: 310) - Feb 18, 2024 - Abstract #USCAP2024USCAP_1150; In urgent cases where CD19 is dim and other markers by flow such as CD79a, CD22 are not uniformly strong, adding PAX5 can "rescue" the leukemia lineage assignment. Recent genome-wide CRISPR screens demonstrate that PAX5 modulates blinatumomab response in B-ALL; possible future directions include studying ways of quantitatively measuring PAX5 expression in these tumors as a predictive marker.
- |||||||||| Ibrance (palbociclib) / Pfizer, Kisqali (ribociclib) / Novartis, Verzenio (abemaciclib) / Eli Lilly
Journal: Therapeutic Monitoring of Palbociclib, Ribociclib, Abemaciclib, M2, M20, and Letrozole in Human Plasma: A Novel LC-MS/MS Method. (Pubmed Central) - Feb 17, 2024 A simple and robust LC-MS/MS method was successfully validated for the simultaneous quantification of CDK4/6is, M2, M20, and letrozole in human plasma. The assay was found to be suitable for measuring steady-state trough concentrations of the analytes in patient samples.
- |||||||||| Journal: Multitarget Potential Drug Candidates for High-Grade Gliomas Identified by Multiple Reaction Monitoring Coupled with In Silico Drug Repurposing. (Pubmed Central) - Feb 16, 2024
The top drug candidates such as Pazopanib, Icotinib, Entrectinib, Regorafenib, and Cabozantinib were explored for their drug-likeness properties using the SwissADME...HGG cell lines showed enhanced cytotoxicity and cell proliferation inhibition with Pazopanib and Temozolomide combinatorial treatment compared to Temozolomide alone...While the present study identified five multitarget-directed potential drug candidates, future clinical studies in larger cohorts are crucial to evaluate the efficacy of these molecular candidates. The research strategy and methodology used in the present study offer new avenues for innovation in drug discovery and development which may prove useful, particularly for cancers with low cure rates.
- |||||||||| Venclexta (venetoclax) / Roche, AbbVie
P1/2 data, Clinical Trial,Phase II, Journal: A Phase 1/2 Study of Mini-Hyper-CVD plus Venetoclax in Patients with Relapsed/Refractory Acute Lymphoblastic Leukemia. (Pubmed Central) - Feb 16, 2024 P1/2 The research strategy and methodology used in the present study offer new avenues for innovation in drug discovery and development which may prove useful, particularly for cancers with low cure rates. Patients received the mini-hyper-CVD regimen (dose-attenuated hyperfractionated cyclophosphamide, vincristine, and dexamethasone alternating with methotrexate and cytarabine) in combination with venetoclax (200
- |||||||||| Repatha (evolocumab) / Amgen, Astellas
Enrollment change, Trial termination: Antiplatelet Effects of Evolocumab in Patients With Peripheral Arterial Disease (clinicaltrials.gov) - Feb 16, 2024 P=N/A, N=30, Terminated, Patients received the mini-hyper-CVD regimen (dose-attenuated hyperfractionated cyclophosphamide, vincristine, and dexamethasone alternating with methotrexate and cytarabine) in combination with venetoclax (200 N=60 --> 30 | Unknown status --> Terminated; Research group transferred to another hospital
- |||||||||| Ibrance (palbociclib) / Pfizer, Erbitux (cetuximab) / Eli Lilly
Trial primary completion date, Metastases: LCCC1717: Palbociclib and Cetuximab in Metastatic Colorectal Cancer (clinicaltrials.gov) - Feb 15, 2024 P2, N=24, Active, not recruiting, Trial primary completion date: Dec 2023 --> Jul 2024 Trial primary completion date: Jan 2026 --> May 2023
- |||||||||| Vectibix (panitumumab) / Amgen
Trial completion date, Trial initiation date, Trial primary completion date: Evaluating 111In Panitumumab for Nodal Staging in Head and Neck Cancer (clinicaltrials.gov) - Feb 15, 2024 P1, N=30, Recruiting, Trial primary completion date: Jan 2024 --> Jul 2024 Trial completion date: Aug 2029 --> Nov 2029 | Initiation date: Dec 2023 --> Apr 2024 | Trial primary completion date: Aug 2028 --> Nov 2028
- |||||||||| carvedilol / Generic mfg., ivabradine / Generic mfg.
Trial completion date, Trial primary completion date: Ivabradine in Cirrhotic Cardiomyopathy (clinicaltrials.gov) - Feb 15, 2024 P=N/A, N=130, Recruiting, Trial completion date: Dec 2023 --> Jun 2024 | Trial primary completion date: Dec 2023 --> Jun 2024 Trial completion date: Dec 2023 --> Dec 2024 | Trial primary completion date: Oct 2023 --> Oct 2024
- |||||||||| Prolia (denosumab) / Amgen
Trial completion date: Denosumab for Smoldering Multiple Myeloma (clinicaltrials.gov) - Feb 15, 2024 P2, N=20, Active, not recruiting, Trial completion date: Dec 2023 --> Dec 2024 | Trial primary completion date: Oct 2023 --> Oct 2024 Trial completion date: Jun 2024 --> Jun 2025
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen, Besponsa (inotuzumab ozogamicin) / Pfizer, UCB
Trial completion date, Trial primary completion date: A041703: Inotuzumab Ozogamicin and Blinatumomab in Treating Patients With Newly Diagnosed, Recurrent, or Refractory CD22-Positive B-Lineage Acute Lymphoblastic Leukemia (clinicaltrials.gov) - Feb 15, 2024 P2, N=64, Recruiting, Trial completion date: Jun 2024 --> Jun 2025 Trial completion date: Feb 2024 --> Feb 2025 | Trial primary completion date: Feb 2024 --> Feb 2025
- |||||||||| Lorbrena (lorlatinib) / Pfizer
Trial completion date, Trial primary completion date: NANT 2015-02: A Phase 1 Study of Lorlatinib (PF-06463922) (clinicaltrials.gov) - Feb 15, 2024 P1, N=65, Active, not recruiting, Trial completion date: Dec 2023 --> Dec 2024 | Trial primary completion date: Dec 2023 --> Dec 2024 Trial completion date: Dec 2024 --> Dec 2025 | Trial primary completion date: Dec 2023 --> Dec 2024
- |||||||||| Ibrance (palbociclib) / Pfizer, gedatolisib (PF-05212384) / Celcuity
Trial completion date, Trial primary completion date, Combination therapy, Metastases: Study of the CDK4/6 Inhibitor Palbociclib (PD-0332991) in Combination With the PI3K/mTOR Inhibitor Gedatolisib (PF-05212384) for Patients With Advanced Squamous Cell Lung, Pancreatic, Head & Neck and Other Solid Tumors (clinicaltrials.gov) - Feb 15, 2024 P1, N=96, Recruiting, Trial completion date: Dec 2024 --> Dec 2025 | Trial primary completion date: Dec 2023 --> Dec 2024 Trial completion date: Jan 2025 --> Jan 2026 | Trial primary completion date: Jan 2024 --> Jan 2025
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