- |||||||||| Ibrance (palbociclib) / Pfizer
Trial completion date, Trial primary completion date, Metastases: Swedish Ibrance Registries Insights (SIRI) (clinicaltrials.gov) - Jun 7, 2024 P=N/A, N=1500, Recruiting, Trial completion date: Dec 2022 --> Aug 2024 | Trial primary completion date: Dec 2022 --> Aug 2024
- |||||||||| dazodalibep (HZN-4920) / Amgen
Enrollment open, Phase classification: VIBRANT: VIB4920 for Active Lupus Nephritis (clinicaltrials.gov) - Jun 6, 2024 P2, N=74, Recruiting, Not yet recruiting --> Recruiting Active, not recruiting --> Recruiting | Phase classification: P2a --> P2
- |||||||||| Ibrance (palbociclib) / Pfizer, Nerlynx (neratinib) / Puma, Lynparza (olaparib) / Merck (MSD), AstraZeneca
Journal, PARP Biomarker: Discovery of acetophenone/piperazin-2-one hybrids as selective anti-TNBC cancer agents by causing DNA damage. (Pubmed Central) - Jun 6, 2024 In addition, 1j could selectively cause DNA damage, inducing the accumulation of ?H2AX and P53 in MDA-MB-468 cells. It also reduced the phosphorylation level of P38 and the expression of HSP70, which further prevented the repair of DNA damage and caused cells S/G2-arrest leading to MDA-MB-468 cells death.
- |||||||||| vepdegestrant (ARV-471) / Arvinas, Pfizer, Ibrance (palbociclib) / Pfizer
Enrollment closed: VERITAC-3: A Study of Vepdegestrant (ARV-471, PF-07850327) Plus Palbociclib Versus Letrozole Plus Palbociclib in Participants With Estrogen Receptor Positive, Human Epidermal Growth Factor Negative Advanced Breast Cancer (clinicaltrials.gov) - Jun 6, 2024 P3, N=1180, Active, not recruiting, These results provide a mechanistic basis for using DS to treat OA. Recruiting --> Active, not recruiting
- |||||||||| palazestrant (OP-1250) / Olema Pharma
Enrollment closed, Enrollment change, Trial completion date, Trial primary completion date, Combination therapy, Metastases: OP-1250-002: A Phase 1 Study of Oral OP-1250 in Combination With Palbociclib in HR+/HER2- Breast Cancer Patients (clinicaltrials.gov) - Jun 6, 2024 P1, N=60, Active, not recruiting, Trial completion date: Aug 2025 --> Aug 2026 | Trial primary completion date: Jan 2025 --> Dec 2025 Recruiting --> Active, not recruiting | N=30 --> 60 | Trial completion date: Dec 2023 --> Jul 2025 | Trial primary completion date: Jan 2023 --> Jan 2025
- |||||||||| Epogen (epoetin alfa) / Amgen
Trial completion, Trial completion date, Trial primary completion date, Adverse events: PAEAN - Erythropoietin for Hypoxic Ischaemic Encephalopathy in Newborns (clinicaltrials.gov) - Jun 4, 2024 P3, N=313, Completed, PCSK9i did not increase neurologic dysfunction, and did not elevate liver enzymes and CK, however it was associated with local injection site reaction. Active, not recruiting --> Completed | Trial completion date: Mar 2023 --> Apr 2024 | Trial primary completion date: Mar 2023 --> Nov 2023
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen
Biomarker, Clinical, Observational data, Retrospective data, Review, Clinical Trial,Phase I, Journal: Pneumocystis jirovecii Pneumonia Secondary to Blinatumomab Therapy: A Case Report. (Pubmed Central) - Jun 4, 2024 Despite prophylaxis, PCP infection cannot be ignored during blinatumomab therapy. Therefore, heightened attention is warranted when using blinatumomab therapy.
- |||||||||| ivabradine / Generic mfg.
Journal: GLP-1 increases heart rate by a direct action on the sinus node. (Pubmed Central) - Jun 4, 2024 GLP-1 has direct chronotropic effects on the heart mediated by GLP-1 receptors in pacemaker cells of the sinus node, inducing changes in action potential morphology and the leading pacemaker site through a calcium signaling response characterized by PKA-dependent phosphorylation of Ca2+ cycling proteins involved in pace making. Targeting the pacemaker calcium clock may be a strategy to lower heart rate in GLP-1 RA recipients.
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen, Darzalex (daratumumab) / J&J, Besponsa (inotuzumab ozogamicin) / Pfizer, UCB
Review, Journal: Naked antibodies and antibody-drug conjugates: targeted therapy for childhood acute lymphoblastic leukemia. (Pubmed Central) - Jun 4, 2024 These antibodies are currently being tested in patients with newly diagnosed ALL and may lead to major changes in the present paradigm of treatment of pediatric ALL. Unlike the past, lessons may be learned from innovations in adult ALL, in which more drastic changes are piloted that may need to be translated to pediatrics.
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen
Review, Journal: Bispecific T-cell engagers in childhood B-acute lymphoblastic leukemia. (Pubmed Central) - Jun 4, 2024 Challenges remain with using BiTE in a broader population although the appeal of now-confirmed reduced toxicity and deeper molecular remissions suggests that this approach will be an essential part of future treatment of childhood B-ALL. Herein, we review some of the pertinent literature covering clinical trials with blinatumomab and address future approaches and combination trials including BiTE.
- |||||||||| Venclexta (venetoclax) / Roche, AbbVie, navtemadlin (KRT-232) / Kartos Therap
Trial completion date, Trial primary completion date, Combination therapy: Testing a New Chemotherapy Drug, KRT-232 (AMG-232) in Combination With Decitabine and Venetoclax in Patients With Acute Myeloid Leukemia (clinicaltrials.gov) - Jun 4, 2024 P1, N=58, Recruiting, Suspended --> Active, not recruiting Trial completion date: Dec 2024 --> Jun 2025 | Trial primary completion date: Dec 2024 --> Jun 2025
- |||||||||| Blincyto (blinatumomab) / Astellas, Amgen
Trial completion date, Trial primary completion date: Lenalidomide and Blinatumomab for the Treatment of Relapsed Non-Hodgkin Lymphoma (clinicaltrials.gov) - Jun 4, 2024 P1, N=44, Active, not recruiting, Trial completion date: Dec 2024 --> Jun 2025 | Trial primary completion date: Dec 2024 --> Jun 2025 Trial completion date: Mar 2025 --> Jun 2025 | Trial primary completion date: Mar 2025 --> Jun 2025
- |||||||||| Jakafi (ruxolitinib) / Incyte, Neupogen (filgrastim) / Kyowa Kirin, Amgen
Journal, Gene Signature: Comprehensive analysis of gene signatures associated with aging in human aortic dissection. (Pubmed Central) - Jun 3, 2024 By sequencing transcriptomic data, this study revealed aging-related hub genes and regulatory network involved in AD formation. Additionally, this study proposed a noteworthy hypothesis that downregulated ESR1 may exacerbate AD by promoting SMC aging, which requires further investigation.
- |||||||||| Simponi (golimumab) / Merck (MSD), Mitsubishi Tanabe, J&J, Cimzia (certolizumab pegol) / Astellas, UCB
Review, Journal: Golimumab and certolizumab pegol for the treatment of hidradenitis suppurativa: a literature review and future perspective. (Pubmed Central) - Jun 3, 2024 (TNF-?) inhibitors, adalimumab, infliximab, and etanercept, are well studied in this patient population, and in some cases, HS was unresponsive to them...Also, golimumab showed promise in treating recalcitrant HS after the failure of other treatments, such as adalimumab and anti-interleukin-1. CPZ and golimumab can be efficacious treatment options for moderate-to-severe HS, especially in patients who are unresponsive to other TNF inhibitors, such as adalimumab.
- |||||||||| Prolia (denosumab) / Amgen
Journal: Denosumab discontinuation: COVID-19 pandemic and beyond. (Pubmed Central) - Jun 3, 2024 However, independent of the "emergency" that occurred during the COVID-19 pandemic, there are other situations in which denosumab is discontinued. In such situations, it is important to have a programmed strategy to optimize care while limiting the risk for unwanted outcomes.
- |||||||||| Journal: Triazole antifungal drug interactions-practical considerations for excellent prescribing. (Pubmed Central) - Jun 2, 2024
We highlight interactions with drugs used in children and new agents introduced for the treatment of haematological malignancies or graft versus host disease (midostaurin, ibrutinib, ruxolitinib and venetoclax). We also summarize the multiple interactions between oral and inhaled corticosteroids and triazole antifungals, and the strategies needed to optimize the therapeutic benefits of triazole antifungal therapy while minimizing potential harm to patients.
- |||||||||| Kepivance (palifermin) / SOBI, Amgen
Journal: Recombinant Human Keratinocyte Growth Factor Ameliorates Cancer Treatment-Induced oral Mucositis on a Chip. (Pubmed Central) - Jun 1, 2024 Palifermin, which is recombinant human keratinocyte growth factor (KGF), is currently the only mitigating treatment available to a subset of OM patients...Cisplatin, radiation, and combined treatments are followed by a recovery period in the OM-OC to determine possible cellular and molecular mechanisms of OM under effects of KGF...Cell damage, barrier dysfunction, and molecular expression during OM induction and resolution were assessed via widefield microscopy, viability and toxicity assays, and antibody arrays. Cell and molecular responses were identified during OM induction and resolution with and without KGF treatment at 1-10
- |||||||||| Imlygic (talimogene laherparepvec) / Amgen
Review, Journal: Cytokine-armed oncolytic herpes simplex viruses: a game-changer in cancer immunotherapy? (Pubmed Central) - Jun 1, 2024 Talimogene laherparepvec is an oncolytic herpes simplex virus type 1 (oHSV), approved for the treatment of recurrent melanoma, and the virus encodes the human cytokine, granulocyte-macrophage colony-stimulating factor (GM-CSF)...In this review, we highlight preliminary data with several cytokines and chemokines, including GM-CSF, interleukin 12, FMS-like tyrosine kinase 3 ligand, tumor necrosis factor ?, interleukin 2, interleukin 15, interleukin 18, chemokine (C-C motif) ligand 2, chemokine (C-C motif) ligand 5, chemokine (C-X-C motif) ligand 4, or their combinations, and show how these payloads can further enhance the antitumor immunity of oHSV. A better understanding of cytokine delivery by oHSV can help improve clinical benefit from oncolytic virus immunotherapy in patients with cancer.
- |||||||||| pasotuxizumab (BAY2010112) / Amgen, Bayer
Inhibition of the de-ubiquitinse USP30 in human fibroblasts from IPF patients suppresses the fibrotic response (PS-6; Poster board no. 13) - May 31, 2024 - Abstract #ERS2024ERS_3796; MTX112 at 10 and 30nM significantly (p<0.05) improved mitochondrial function by 50% in IPF fibroblasts. Targeting USP30 may therefore be a novel therapeutic strategy for the treatment of pulmonary fibrosis by improving pulmonary fibroblast mitochondrial function and slowing tissue fibrosis, potentially halting disease progression.
- |||||||||| Tezspire (tezepelumab-ekko) / AstraZeneca, Amgen
Tezepelumab reduces the expression of MUC5AC in patients with asthma (A1) - May 31, 2024 - Abstract #ERS2024ERS_3516; Anti-TSLP treatment reduces the expression of MUC5AC independent of T2-biomarker status, possibly through a downregulation of the EGFR pathway. This could mechanistically explain how tezepelumab reduces mucus plugging.
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