- |||||||||| Afinitor (everolimus) / Novartis
Journal, Combination therapy: Everolimus in combination with Imatinib overcomes resistance in Chronic myeloid leukaemia. (Pubmed Central) - Jun 15, 2019 The response to Everolimus was influenced by TKI treatment, with a better response in samples from patients under 2nd and 3rd generation TKI and with less toxicity to lymphocytes. Our results reveal that Everolimus induce cell death in CML cells sensitive and resistant to Imatinib, with low cytotoxicity to normal cells, suggesting that Everolimus could be an alternative targeted therapeutic approach in CML patients, even in cases of Imatinib resistance.
- |||||||||| Afinitor (everolimus) / Novartis
Clinical, Journal: Long-Term Clinical and Angiographic Outcomes After Implantation of New-Generation Drug-Eluting Stents for Patients on Maintenance Hemodialysis. (Pubmed Central) - Jun 14, 2019 ...This study aims to investigate the long-term clinical and angiographic outcomes after new-generation DES implantation for hemodialysis patients.We retrospectively enrolled 91 consecutive patients (118 lesions) who underwent successful new-generation DES (everolimus-, zotarolimus-, and biolimus-eluting stents) implantation for the first time...The serum calcium level was significantly higher in the MACCE group (9.34 ± 0.92 mg/dL versus 8.77 ± 0.88 mg/dL; P = 0.004). The multivariate Cox proportional hazards model revealed that the serum calcium level (hazard ratio, 1.86; 95% confidence interval [CI]: 1.26-2.77; P = 0.002), suboptimal (over 55 mg/dL) calcium-phosphorus product (hazard ratio, 3.27; 95% CI: 1.41-7.61; P = 0.006) and the coexistence of peripheral artery disease (hazard ratio, 3.15; 95% CI: 1.49-6.65; P = 0.003) were independent predictors of MACCE.For hemodialysis patients, MACCE remains a frequent occurrence after new-generation DES implantation and is associated with calcium-phosphate metabolism and peripheral artery disease.
- |||||||||| Campath (alemtuzumab) / Sanofi, Afinitor (everolimus) / Novartis
Review, Journal: Novel and Future Therapeutic Drugs for Advanced Mycosis Fungoides and Sézary Syndrome. (Pubmed Central) - Jun 14, 2019 This review provides a discussion of the recent and future promising therapeutic approaches in the management of advanced MF/SS. These include mogamulizumab, brentuximab vedotin, alemtuzumab, immune checkpoint inhibitors, IPH4102 (anti-KIR3DL2 antibody), histone deacetylase inhibitors (vorinostat, romidepsin, panobinostat, belinostat, and resminostat), pralatrexate, forodesine, denileukin diftitox, duvelisib, lenalidomide, and everolimus.
- |||||||||| Imbruvica (ibrutinib) / AbbVie, J&J
Enrollment change, Trial completion date, Trial primary completion date, Combination therapy, Metastases: Study to Evaluate Ibrutinib Combination Therapy in Patients With Selected Gastrointestinal and Genitourinary Tumors (clinicaltrials.gov) - Jun 12, 2019 P1b/2, N=348, Recruiting, These include mogamulizumab, brentuximab vedotin, alemtuzumab, immune checkpoint inhibitors, IPH4102 (anti-KIR3DL2 antibody), histone deacetylase inhibitors (vorinostat, romidepsin, panobinostat, belinostat, and resminostat), pralatrexate, forodesine, denileukin diftitox, duvelisib, lenalidomide, and everolimus. N=261 --> 348 | Trial completion date: Jun 2019 --> May 2021 | Trial primary completion date: Feb 2019 --> May 2021
- |||||||||| Taltorvic (ridaforolimus) / Takeda, Merck (MSD), Afinitor (everolimus) / Novartis
Journal: The EluNIR Ridaforolimus Eluting Coronary Stent System. (Pubmed Central) - Jun 9, 2019 The stent has thin struts with variable widths and a delivery catheter with a spring tip. These characteristics may explain the good angiographic and clinical results of this stent, which were non-inferior to the FDA approved Medtronic Resolute stent DES.
- |||||||||| Sutent (sunitinib) / Pfizer
Trial completion date, Trial primary completion date, Metastases: Potential Molecular Predictors of Response to Novel Therapies in Metastatic Pancreatic Neuroendocrine Tumors (clinicaltrials.gov) - Jun 4, 2019 P=N/A, N=30, Recruiting, Our limited single center experience shows encouraging response to use of somatostatin analogs, azithromycin, and everolimus in the management of debilitating DIPNECH associated symptoms. Trial completion date: May 2019 --> May 2020 | Trial primary completion date: May 2019 --> May 2020
- |||||||||| everolimus / Generic mfg.
Preclinical, Journal: In Vivo Evaluation of Dual-Targeted Nanoparticles Encapsulating Paclitaxel and Everolimus. (Pubmed Central) - May 31, 2019 While maintaining anti-tumor efficacy, the levels of body weight loss were significantly lower (p < 0.0001) and the overall degree of neurotoxicity was reduced with Dual-NP treatment in comparison to the free-drug combination when administered at an equivalent dose of PTX. This study suggests that Dual-NPs present a promising platform for the delivery of the PTX and EVER combination with the potential to reduce severe PTX-induced toxicities and in turn, improve quality of life for patients with BC.
- |||||||||| everolimus / Generic mfg.
Trial completion date, Trial primary completion date, Combination therapy, Metastases: Everolimus Combined With Anti-estrogen Therapy in Hormone-Receptor-Positive HER-2 Negative Advanced Breast Cancer (clinicaltrials.gov) - May 30, 2019 P2, N=48, Active, not recruiting, This study suggests that Dual-NPs present a promising platform for the delivery of the PTX and EVER combination with the potential to reduce severe PTX-induced toxicities and in turn, improve quality of life for patients with BC. Trial completion date: Jan 2019 --> Jan 2020 | Trial primary completion date: Jan 2019 --> Jan 2020
- |||||||||| Afinitor (everolimus) / Novartis
Clinical, Clinical data, Journal: Primary hepatic angiosarcoma and liver transplantation: Radiological, surgical, histological findings and clinical outcome. (Pubmed Central) - May 30, 2019 Because of the histological findings, tacrolimus was switched to everolimus as the main immunosuppressive drug one month after LT...Consequently, HAS remains an absolute contraindication to LT because of the poor outcome. If LT has been performed for incidental HAS, new molecular therapies (e.g. vascular endothelial growth factor antagonists) should be considered immediately after LT to improve the outcome.
- |||||||||| Afinitor (everolimus) / Novartis
Review, Journal: Renal Protection Strategies after Heart Transplantation. (Pubmed Central) - May 30, 2019 This review outlines the recent results of using these renal protection strategies including their drawbacks. We also discuss alternative approaches to optimized individual immunosuppressive therapies after HTx.
- |||||||||| metformin / Generic mfg., everolimus / Generic mfg., exemestane / Generic mfg.
Enrollment change, Metastases: Exemestane-RAD001-Metformin (clinicaltrials.gov) - May 29, 2019 P2, N=23, Terminated, Treatment with mTOR inhibitors can reverse graft dysfunction in approximately half of patients. N=40 --> 23
- |||||||||| everolimus / Generic mfg.
Biomarker, Review, Journal: Targeting the PI3K pathway in cancer: are we making headway? (Pubmed Central) - May 24, 2019 Finally, considering that oncogenic activation of the PI3K-AKT-mTOR pathway often occurs alongside pro-tumorigenic aberrations in other signalling networks, rational combinations are also needed to optimize the effectiveness of treatment. Herein, we review the current experience with anticancer therapies that target the PI3K-AKT-mTOR pathway.
- |||||||||| everolimus / Generic mfg.
Enrollment closed, Metastases: Phase IV Study of the Safety and Efficacy of Everolimus in Adult Patients With Progressive pNET in China (clinicaltrials.gov) - May 24, 2019 P4, N=49, Active, not recruiting, Although the comprehensive immunomonitoring analysis performed in this study provides relevant information for the design of future immunotherapeutic approaches, the addition of metronomic cyclophosphamide to mRCC patients receiving everolimus cannot be recommended. Recruiting --> Active, not recruiting
- |||||||||| Afinitor (everolimus) / Novartis, Opdivo (nivolumab) / Ono Pharma, BMS
Clinical, Journal: Management of relapsed/refractory classical Hodgkin lymphoma in transplant-ineligible patients. (Pubmed Central) - May 15, 2019 For patients who have failed prior transplant or are unsuitable for dose-intense approaches based on age or comorbidities, an individualized approach with sequential use of single agents such as brentuximab vedotin, PD-1 inhibitors, everolimus, lenalidomide, or conventional agents such as gemcitabine or vinorelbine, may result in prolonged survivals with minimal or modest effect on quality of life. Participation in clinical trials evaluating new approaches such as combination immune checkpoint inhibition, novel antibody-drug conjugates, or cellular therapies such as EBV-directed cytotoxic T-lymphocytes and chimeric antigen receptor T-cells offer additional options for eligible patients.
- |||||||||| Afinitor (everolimus) / Novartis
Journal: 2-Oxonanonoidal Antibiotic Actinolactomycin Inhibits Cancer Progression by Suppressing HIF-1α. (Pubmed Central) - May 15, 2019 More interestingly, low dose of ALM treatment enhanced the anti-tumor effect of Everolimus, an inhibitor of mTOR, suggesting its potential use in combination therapy of tumors, especially solid tumor patients. Thus, we identified a novel HIF-1α inhibitor from the metabolites of Streptomyces flavoretus, which shows promising anti-cancer potential.
- |||||||||| Zolinza (vorinostat) / Merck (MSD), Torisel (temsirolimus) / Pfizer
Trial completion date, Trial primary completion date, Epigenetic controller, Metastases: Sirolimus or Everolimus or Temsirolimus and Vorinostat in Advanced Cancer (clinicaltrials.gov) - May 15, 2019 P1, N=249, Active, not recruiting, Trial completion date: Sep 2019 --> Sep 2020 Trial completion date: Mar 2019 --> May 2021 | Trial primary completion date: Mar 2019 --> May 2020
|