- |||||||||| Yondelis (trabectedin) / Otsuka, PharmaMar, Valeo Pharma, Zepzelca (lurbinectedin) / PharmaMar, Jazz
Journal: A scalable total synthesis of Et-743 and lurbinectedin. (Pubmed Central) - Aug 30, 2020 Thus, the clinical activity of lurbinectedin may originate, at least in part, from the induction of ICD. An efficient and scalable approach for total synthesis of Et-743 and lubinectedin (about 1.6% overall yield in 26 total steps from Cbz-protected (S)-tyrosine) is described, and features the use of a common advanced intermediate to create the right and left parts of these antitumor drugs, and a light-mediated remote C-H bond activation to assemble a benzo[1,3]dioxole-embodied intermediate.
- |||||||||| Zepzelca (lurbinectedin) / PharmaMar, Jazz
Vamos ZepZelCa 👍👏👏 (Twitter) - Aug 5, 2020
- |||||||||| doxorubicin hydrochloride / Generic mfg., Zepzelca (lurbinectedin) / PharmaMar, Jazz
Clinical, P2 data, Journal, Pan Tumor: Lurbinectedin as second-line treatment for patients with small-cell lung cancer: a single-arm, open-label, phase 2 basket trial. (Pubmed Central) - Jul 10, 2020 P2 Lurbinectedin was active as second-line therapy for SCLC in terms of overall response and had an acceptable and manageable safety profile. Lurbinectedin could represent a potential new treatment for patients with SCLC, who have few options especially in the event of a relapse, and is being investigated in combination with doxorubicin as second-line therapy in a randomised phase 3 trial.
- |||||||||| Zepzelca (lurbinectedin) / PharmaMar, Jazz
Zepzelca (Twitter) - Jun 18, 2020
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