molibresib (GSK525762) / GSK  >>  Phase 2
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5 Trials

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Trial + Data / EventsStatusPhNRegionInterventionsSponsorConditionsPrimary complStudy compl
molibresib (GSK525762) / GSK
NCT01943851: A Dose Escalation Study to Investigate the Safety, Pharmacokinetics (PK), Pharmacodynamics (PD) and Clinical Activity of GSK525762 in Subjects With Relapsed, Refractory Hematologic Malignancies

Hourglass Jul 2020 - Dec 2020 : In hematologic malignancies
Checkmark Initiation of expansion cohorts in P1 trial in hematologic malignancies
Jun 2017 - Jun 2017: Initiation of expansion cohorts in P1 trial in hematologic malignancies
Completed
2
111
Europe, US, RoW
GSK525762
GlaxoSmithKline
Neoplasms
04/20
04/20
NCT03266159: A Dose Escalation Study to Investigate the Safety, Pharmacokinetics (PK), Pharmacodynamics (PD), and Clinical Activity of GSK525762 Plus Trametinib in Subjects With Solid Tumors

Withdrawn
2
0
NA
GSK525762 Besylate tablets, Trametinib tablets
GlaxoSmithKline
Solid Tumours
08/20
08/20
NCT01587703 / 2014-004982-25: A Study to Investigate the Safety, Pharmacokinetics, Pharmacodynamics, and Clinical Activity of GSK525762 in Subjects With NUT Midline Carcinoma (NMC) and Other Cancers

Completed
1/2
196
Europe, US, RoW
GSK525762
GlaxoSmithKline
Carcinoma, Midline
04/18
07/19
NCT04116359: Testing of the Addition of a New Anti-cancer Drug, Molibresib, to Chemotherapy Treatment (Etoposide and Cisplatin) for Patients With NUT Carcinoma

Withdrawn
1/2
0
NA
Cisplatin, Abiplatin, Blastolem, Briplatin, CDDP, Cis-diammine-dichloroplatinum, Cis-diamminedichloridoplatinum, Cis-diamminedichloro Platinum (II), Cis-diamminedichloroplatinum, Cis-dichloroammine Platinum (II), Cis-platinous Diamine Dichloride, Cis-platinum, Cis-platinum II, Cis-platinum II Diamine Dichloride, Cismaplat, Cisplatina, Cisplatinum, Cisplatyl, Citoplatino, Citosin, Cysplatyna, DDP, Lederplatin, Metaplatin, Neoplatin, Peyrone''s Chloride, Peyrone''s Salt, Placis, Plastistil, Platamine, Platiblastin, Platiblastin-S, Platinex, Platinol, Platinol- AQ, Platinol-AQ, Platinol-AQ VHA Plus, Platinoxan, Platinum, Platinum Diamminodichloride, Platiran, Platistin, Platosin, Etoposide, Demethyl Epipodophyllotoxin Ethylidine Glucoside, EPEG, Lastet, Toposar, Vepesid, VP 16, VP 16-213, VP-16, VP-16-213, VP16, Etoposide Phosphate, Etopophos, Molibresib, GSK-525762A, GSK525762, I-BET 762, Molibresib Besylate, GSK525762C
National Cancer Institute (NCI)
Metastatic NUT Carcinoma, Unresectable NUT Carcinoma
09/20
09/20
NCT02964507 / 2016-003074-40: Dose Escalation and Expansion Study of GSK525762 in Combination With Fulvestrant in Participants With Hormone Receptor-positive (HR+)/Human Epidermal Growth Factor Receptor 2 Negative (HER2-) Advanced or Metastatic Breast Cancer

Hourglass Feb 2020 - Jun 2020 : Proof-of-concept data from trial for ER+ breast cancer
Terminated
1/2
124
Europe, Canada, US, RoW
GSK525762, Placebo, Fulvestrant
GlaxoSmithKline
Neoplasms
09/20
07/21

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