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Kinase Inhibitors
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Phase 2
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berzosertib
(M6620) / EMD Serono
peposertib
(M3814) / EMD Serono
samotolisib
(LY3023414) / Eli Lilly
ulixertinib
(BVD-523) / BioMed Valley Discoveries
tuvusertib
(M1774) / EMD Serono
refametinib
(BAY86-9766) / Bayer
zimlovisertib
(PF-06650833) / Pfizer
temuterkib
(LY3214996) / Eli Lilly
Hocena
(antroquinonol) / Golden Biotechnology
elimusertib
(BAY 1895344) / Bayer
emavusertib
(CA-4948) / Curis, Dr. Reddy’s
GSK2982772
/ GSK
amcasertib
(BBI-503) / Sumitomo Pharma
oditrasertib
(DNL788) / Denali Therap, Sanofi
LP-168
/ Lupeng Pharma
PXL770
/ Poxel SA
camonsertib
(RP-3500) / Repare Therap
itanapraced
(CHF-5074) / CereSpir
zabedosertib
(BAY 1834845) / Bayer
vutiglabridin
(HSG4112) / Glaceum
ASN007
/ Asana BioSci, Erasca, UT MD Anderson Cancer Center
BI 706321
/ Boehringer Ingelheim
CBP501
/ CanBas
edecesertib
(GS-5718) / Gilead
ocadusertib
(LY3871801) / Eli Lilly
rineterkib
(LTT462) / Novartis
ASTX029
/ Otsuka
SF1126
/ SignalRx
ART0380
/ Artios Pharma
AZD7648
/ AstraZeneca
GFH312
/ GenFleet Therap
JTT-251
/ Japan Tobacco
SAR444656
/ Sanofi
SC0245
/ Shijiazhuang Sagacity, Wuxi Biocity
eclitasertib
(DNL758) / Denali Therap, Sanofi
gartisertib
(M4344) / EMD Serono
simurosertib
(TAK-931) / Takeda, ZAI Lab
ABBV-668 IR
/ AbbVie
DCC-3116
/ Ono Pharma
DTRM-555
/ Zhejiang DTRM Biopharma
H-1337
/ D. Western Therapeutics Institute
HRS2398
/ Jiangsu Hengrui Pharma
LM-061
/ LaNova Medicines Limited
TQH3821
/ Sino Biopharm
leucine/metformin/sildenafil
(NS-0200) / NuSirt
tanzisertib
(CC 930) / BMS
AEG33773
/ Pharmascience
ASP1570
/ Astellas
ATRN-119
/ Aprea
C019199
/ Fujian Haixi New Pharmaceutical
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