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Phase
N/A
1
2
3
4
Trials
0
7
14
21
28
35
42
49
56
63
70
adavosertib
(AZD1775) / AstraZeneca
ZEN-3694
/ Zenith Capital Corp
azenosertib
(ZN-c3) / Zentalis Pharma
Ezharmia
(valemetostat) / Daiichi Sankyo
davamotecan pegadexamer
(EP0057) / Ellipses Pharma
rocilinostat
(ACY-1215) / Regenacy
BI2536
/ Boehringer Ingelheim
foscenvivint
(PRI724) / PRISM Pharma, Ohara Pharma
diclostat
(BEBT-908) / BeBetter Med
domatinostat
(4SC-202) / 4SC
firtecan pegol
(PEG-SN38) / Belrose
iadademstat
(ORY-1001) / Oryzon
molibresib
(GSK525762) / GSK
vafidemstat
(ORY-2001) / Oryzon
E7386
/ Eisai, PRISM Pharma
tinostamustine
(EDO-S101) / Mundipharma
FX 322
/ Astellas, Korro Bio
OPN-2853
/ Opna Bio
decitabine/ tetrahydrouridine
(EPI01) / EpiDestiny, Novo Nordisk
fimepinostat
(CUDC-907) / Curis
nanatinostat
(VRx-3996) / Viracta Therap
Lipotecan
(TLC388) / Taiwan Liposome Company
Rezlidhia
(olutasidenib) / Rigel
SRA515
/ GSK
birabresib
(OTX015) / Merck (MSD)
ivaltinostat IV
(CG-745) / CG Invites
quisinostat
(JNJ 26481585) / ChemRar, Viriom
safusidenib
(DS-1001) / Daiichi Sankyo, Nuvation Bio
CUDC-101
/ Curis
Debio 0123
/ Debiopharm
MK-3795
/ Merck (MSD)
Sulforadex
(sulforafan alfadex) / Evgen Pharma, STALICLA
ezobresib
(BMS-986158) / BMS
panobinostat
(MTX110) / Biodexa Pharma
pulrodemstat
(CC-90011) / BMS
remetinostat
(SHP-141) / Medivir
seclidemstat
(SP2577) / Salarius
zabinostat
(CXD101) / IngenOx Therap, Nuance Biotech
AMG 193
/ Amgen
IDH305
/ Novartis
INCB59872
/ Incyte
NKT2152
/ NiKang Therap
QN-165
/ Qualigen Therap
SF1126
/ SignalRx
casdatifan
(AB521) / Arcus Biosci
etrinabdione
(EHP-101) / Emerald Health Pharmaceuticals, Aphios, Emerald Health Research
pinometostat
(EPZ-5676) / Ipsen
CKD-506
/ Chong Kun Dang
GB004
/ Aadi Biosci
GSK2879552
/ GSK
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