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Serine-Threonine Kinase Inhibitors
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Phase
N/A
1
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Trials
0
99
198
297
396
495
594
693
792
891
990
ENMD-2076
/ CASI
GLPG3970
/ Galapagos, Gilead
MK-1084
/ Merck (MSD)
QTORIN 3.9%
(rapamycin topical) / Palvella Therapeutics
SPH4336
/ Shanghai Pharma
fadraciclib
(CYC065) / Cyclacel
miransertib
(MK-7075) / Merck (MSD)
seliciclib
(CYC202) / Cyclacel, Cedars-Sinai
zotiraciclib
(TG02) / Cothera Biosci
AZD1390
/ AstraZeneca
FX 322
/ Astellas, Korro Bio
RVU120
/ Ryvu Therap
VIC-1911
/ VITRAC Therap
barasertib-HQPA
(AZD2811) / AstraZeneca
milciclib
(TZLS-201) / Tiziana Life Sci
naporafenib
(ERAS-254) / Erasca
niclosamide topical
(ATx 201) / UNION Therap
ocifisertib
(CFI-400945) / Treadwell Therap
pembrolizumab/berahyaluronidase alfa
(MK-3475A) / Merck (MSD)
phenoxodiol
(NV06) / MEI
sonolisib
(PX 866) / Pfizer
tigilanol tiglate
(EBC-46) / Qbiotics
AL8326
/ Advenchen
AT9283
/ Otsuka
BI 1701963
/ Boehringer Ingelheim
CINelim
(terameprocol) / Erimos Pharma
E6201
/ Strategia Therap
bireociclib
(XZP 3287) / Sihuan Pharmaceutical
ibrilatazar
(ABTL0812) / Ability Pharma
plixorafenib
(FORE-8394) / Fore Biotherap
sitneprotafib
(JAB-3312) / Jacobio Pharma
zilurgisertib
(INCB00928) / Incyte
AT7519
/ Novartis, Otsuka
AZD8055
/ AstraZeneca
ERAS-007
/ Erasca
ETP-47187
/ CNIO
Fantom
(sirolimus-eluting bioresorbable scaffold) / REVA Medical
MS-553
/ MingSight Pharma
PF-04691502
/ Pfizer
Rapalimus Gel
(sirolimus gel) / Nobelpharma
SEL-110
/ Cartesian Therap
SPN-820
/ Navitor Pharma, Supernus Pharma
WXFL10030390
/ Guangzhou JOYO Pharma
Zonalta
(Z-endoxifen hydrochloride) / Jina Pharma, Intas
belvarafenib
(RG6185) / Hanmi
bryostatin 1
(NSC 339555) / Synaptogenix
danusertib
(PHA-739358) / Nerviano Medical Sciences
darovasertib
(IDE196) / Ideaya Biosci
narazaciclib
(HX301) / Traws Pharma
niclosamide
(DWRX2003) / Daewoong Pharma
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