Serine-Threonine Kinase Inhibitors 

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ENMD-2076 / CASI           
          
            
             
GLPG3970 / Galapagos, Gilead           
          
            
             
MK-1084 / Merck (MSD)           
          
            
             
QTORIN 3.9% (rapamycin topical) / Palvella Therapeutics           
          
            
             
SPH4336 / Shanghai Pharma           
          
            
             
fadraciclib (CYC065) / Cyclacel           
          
            
             
miransertib (MK-7075) / Merck (MSD)           
          
            
             
seliciclib (CYC202) / Cyclacel, Cedars-Sinai           
          
            
             
zotiraciclib (TG02) / Cothera Biosci           
          
            
             
AZD1390 / AstraZeneca           
          
            
             
FX 322 / Astellas, Korro Bio           
          
            
             
RVU120 / Ryvu Therap           
          
            
             
VIC-1911 / VITRAC Therap           
          
            
             
barasertib-HQPA (AZD2811) / AstraZeneca           
          
            
             
milciclib (TZLS-201) / Tiziana Life Sci           
          
            
             
naporafenib (ERAS-254) / Erasca           
          
            
             
niclosamide topical (ATx 201) / UNION Therap           
          
            
             
ocifisertib (CFI-400945) / Treadwell Therap           
          
            
             
pembrolizumab/berahyaluronidase alfa (MK-3475A) / Merck (MSD)           
          
            
             
phenoxodiol (NV06) / MEI           
          
            
             
sonolisib (PX 866) / Pfizer           
          
            
             
tigilanol tiglate (EBC-46) / Qbiotics           
          
            
             
AL8326 / Advenchen           
          
            
             
AT9283 / Otsuka           
          
            
             
BI 1701963 / Boehringer Ingelheim           
          
            
             
CINelim (terameprocol) / Erimos Pharma           
          
            
             
E6201 / Strategia Therap           
          
            
             
bireociclib (XZP 3287) / Sihuan Pharmaceutical           
          
            
             
ibrilatazar (ABTL0812) / Ability Pharma           
          
            
             
plixorafenib (FORE-8394) / Fore Biotherap           
          
            
             
sitneprotafib (JAB-3312) / Jacobio Pharma           
          
            
             
zilurgisertib (INCB00928) / Incyte           
          
            
             
AT7519 / Novartis, Otsuka           
          
            
             
AZD8055 / AstraZeneca           
          
            
             
ERAS-007 / Erasca           
          
            
             
ETP-47187 / CNIO           
          
            
             
Fantom (sirolimus-eluting bioresorbable scaffold) / REVA Medical           
          
            
             
MS-553 / MingSight Pharma           
          
            
             
PF-04691502 / Pfizer           
          
            
             
Rapalimus Gel (sirolimus gel) / Nobelpharma           
          
            
             
SEL-110 / Cartesian Therap           
          
            
             
SPN-820 / Navitor Pharma, Supernus Pharma           
          
            
             
WXFL10030390 / Guangzhou JOYO Pharma           
          
            
             
Zonalta (Z-endoxifen hydrochloride) / Jina Pharma, Intas           
          
            
             
belvarafenib (RG6185) / Hanmi           
          
            
             
bryostatin 1 (NSC 339555) / Synaptogenix           
          
            
             
danusertib (PHA-739358) / Nerviano Medical Sciences           
          
            
             
darovasertib (IDE196) / Ideaya Biosci           
          
            
             
narazaciclib (HX301) / Traws Pharma           
          
            
             
niclosamide (DWRX2003) / Daewoong Pharma           
          
            
            


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