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Serine-Threonine Kinase Inhibitors
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Phase
N/A
1
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Trials
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99
198
297
396
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693
792
891
990
vactosertib
(TEW-7197) / National OncoVenture, Theragen Etex
dinaciclib
(MK-7965) / Merck (MSD)
niclosamide
/ Generic mfg.
ulixertinib
(BVD-523) / BioMed Valley Discoveries
chiauranib
(CS 2164) / Chipscreen
samotolisib
(LY3023414) / Eli Lilly
culmerciclib
(TQB3616) / Sino Biopharm
Arxxant
(ruboxistaurin oral) / Eli Lilly, Takeda
LY3295668
/ Eli Lilly
Ojemda
(tovorafenib) / Day One Biopharma
onvansertib
(PCM-075) / Cardiff Oncology
paxalisib
(GDC-0084) / Kazia, SoVarGen, QIMR Berghofer Medical Research Institute
Opsiria
(sirolimus) / Santen
refametinib
(BAY86-9766) / AstraZeneca
uprosertib
(LAE003) / Laekna Therap
Nypta
(tideglusib) / ASD Therap
RX208
/ Suzhou NeuPharma
ST266
/ Noveome Biotherap
apitolisib
(GDC-0980) / Roche
divarasib
(RG6330) / Roche
fovinaciclib
(FCN-437) / Fosun Pharma
glecirasib
(JAB-21822) / Jacobio Pharma
riviciclib
(P27600) / Piramal Phytocare
BI2536
/ Boehringer Ingelheim
HRS-4642
/ Jiangsu Hengrui Pharma
Relyvrio
(phenylbutyrate/taurursodiol) / Amylyx
Triolex
(bezisterim) / BioVie
atirmociclib
(PF-07220060) / Pfizer
bimiralisib
(PQR309) / Torqur
elraglusib
(9-ING-41) / Actuate Therap
indisulam
(E7070) / Eisai
olomorasib
(LY3537982) / Eli Lilly
omipalisib
(GSK2126458) / GSK
temuterkib
(LY3214996) / Eli Lilly
voxtalisib
(SAR245409) / Sanofi
Hocena
(antroquinonol) / Golden Biotechnology
fezagepras
(PBI-4050) / Liminal BioSci
garsorasib
(D-1553) / InventisBio
onatasertib
(ATG-008) / BMS
opnurasib
(JDQ443) / Novartis
silmitasertib
(CX-4945) / Senhwa Biosci
tinengotinib
(TT-00420) / TransThera Biosci
barasertib
(AZD1152) / AstraZeneca
lerociclib
(G1T38) / Walvax, Pepper Bio
polyinosinic:polycytidylic acid
(BO-112) / Highlight Therap
roniciclib
(BAY1000394) / Bayer
tomivosertib
(eFT508) / eFFECTOR Therap
tozasertib
(MK-0457) / Merck (MSD)
BEBT-209
/ BeBetter Med
Dupert
(fulzerasib) / GenFleet Therap
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