Serine-Threonine Kinase Inhibitors 

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vactosertib (TEW-7197) / National OncoVenture, Theragen Etex           
          
            
             
dinaciclib (MK-7965) / Merck (MSD)           
          
            
             
niclosamide / Generic mfg.           
          
            
             
ulixertinib (BVD-523) / BioMed Valley Discoveries           
          
            
             
chiauranib (CS 2164) / Chipscreen           
          
            
             
samotolisib (LY3023414) / Eli Lilly           
          
            
             
culmerciclib (TQB3616) / Sino Biopharm           
          
            
             
Arxxant (ruboxistaurin oral) / Eli Lilly, Takeda           
          
            
             
LY3295668 / Eli Lilly           
          
            
             
Ojemda (tovorafenib) / Day One Biopharma           
          
            
             
onvansertib (PCM-075) / Cardiff Oncology           
          
            
             
paxalisib (GDC-0084) / Kazia, SoVarGen, QIMR Berghofer Medical Research Institute           
          
            
             
Opsiria (sirolimus) / Santen           
          
            
             
refametinib (BAY86-9766) / AstraZeneca           
          
            
             
uprosertib (LAE003) / Laekna Therap           
          
            
             
Nypta (tideglusib) / ASD Therap           
          
            
             
RX208 / Suzhou NeuPharma           
          
            
             
ST266 / Noveome Biotherap           
          
            
             
apitolisib (GDC-0980) / Roche           
          
            
             
divarasib (RG6330) / Roche           
          
            
             
fovinaciclib (FCN-437) / Fosun Pharma           
          
            
             
glecirasib (JAB-21822) / Jacobio Pharma           
          
            
             
riviciclib (P27600) / Piramal Phytocare           
          
            
             
BI2536 / Boehringer Ingelheim           
          
            
             
HRS-4642 / Jiangsu Hengrui Pharma           
          
            
             
Relyvrio (phenylbutyrate/taurursodiol) / Amylyx           
          
            
             
Triolex (bezisterim) / BioVie           
          
            
             
atirmociclib (PF-07220060) / Pfizer           
          
            
             
bimiralisib (PQR309) / Torqur           
          
            
             
elraglusib (9-ING-41) / Actuate Therap           
          
            
             
indisulam (E7070) / Eisai           
          
            
             
olomorasib (LY3537982) / Eli Lilly           
          
            
             
omipalisib (GSK2126458) / GSK           
          
            
             
temuterkib (LY3214996) / Eli Lilly           
          
            
             
voxtalisib (SAR245409) / Sanofi           
          
            
             
Hocena (antroquinonol) / Golden Biotechnology           
          
            
             
fezagepras (PBI-4050) / Liminal BioSci           
          
            
             
garsorasib (D-1553) / InventisBio           
          
            
             
onatasertib (ATG-008) / BMS           
          
            
             
opnurasib (JDQ443) / Novartis           
          
            
             
silmitasertib (CX-4945) / Senhwa Biosci           
          
            
             
tinengotinib (TT-00420) / TransThera Biosci           
          
            
             
barasertib (AZD1152) / AstraZeneca           
          
            
             
lerociclib (G1T38) / Walvax, Pepper Bio           
          
            
             
polyinosinic:polycytidylic acid (BO-112) / Highlight Therap           
          
            
             
roniciclib (BAY1000394) / Bayer           
          
            
             
tomivosertib (eFT508) / eFFECTOR Therap           
          
            
             
tozasertib (MK-0457) / Merck (MSD)           
          
            
             
BEBT-209 / BeBetter Med           
          
            
             
Dupert (fulzerasib) / GenFleet Therap           
          
            
            


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