Serine-Threonine Kinase Inhibitors 

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 Trials
 097194291388485582679776873970
            
            
             
sorafenib / Generic mfg.           
          
            
             
everolimus / Generic mfg.           
          
            
             
sirolimus / Generic mfg.           
          
            
             
Ibrance (palbociclib) / Pfizer           
          
            
             
Stivarga (regorafenib) / Bayer           
          
            
             
Votrient (pazopanib) / Novartis, BeiGene           
          
            
             
Xience (everolimus-eluting stent) / Abbott           
          
            
             
Epidaza (chidamide) / Chipscreen, Meiji Seika, Eisai, HUYA Bioscience           
          
            
             
Torisel (temsirolimus) / Pfizer           
          
            
             
Verzenio (abemaciclib) / Eli Lilly           
          
            
             
Tafinlar (dabrafenib) / Novartis, BeiGene           
          
            
             
Zelboraf (vemurafenib) / Roche           
          
            
             
Kisqali (ribociclib) / Novartis           
          
            
             
Viracept (nelfinavir) / ViiV Healthcare, Roche           
          
            
             
Resolute ZES (zotarolimus-eluting stent) / Medtronic           
          
            
             
AiRuiKang (dalpiciclib) / Jiangsu Hengrui Pharma           
          
            
             
Braftovi (encorafenib) / Ono Pharma, Pierre Fabre, Pfizer           
          
            
             
Zepsun (donafenib) / Suzhou Zelgen           
          
            
             
ingenol mebutate / Generic mfg.           
          
            
             
Lumakras (sotorasib) / Amgen           
          
            
             
alvocidib (DSP-2033) / Sumitomo Pharma           
          
            
             
alisertib (MLN8237) / Puma           
          
            
             
ipatasertib (RG7440) / Roche           
          
            
             
Rydapt (midostaurin) / Novartis           
          
            
             
Truqap (capivasertib) / Otsuka, AstraZeneca           
          
            
             
Kinenza (enzastaurin) / Denovo, Aytu BioPharma           
          
            
             
MK-2206 / Merck (MSD)           
          
            
             
ceralasertib (AZD6738) / AstraZeneca           
          
            
             
Vonjo (pacritinib) / SOBI           
          
            
             
Taltorvic (ridaforolimus) / Takeda, Merck (MSD)           
          
            
             
sapanisertib (CB-228) / Calithera           
          
            
             
perifosine (D21266) / AEterna Zentaris           
          
            
             
dordaviprone (ONC201) / Chimerix           
          
            
             
vistusertib (AZD2014) / AstraZeneca           
          
            
             
Estybon (rigosertib) / Onconova, SymBio Pharma, Knight Therap           
          
            
             
retlirafusp alfa (SHR-1701) / Jiangsu Hengrui Pharma           
          
            
             
Ukoniq (umbralisib) / TG Therap           
          
            
             
Absorb (everolimus-eluting bioresorbable vascular scaffold) / Abbott           
          
            
             
Turalio (pexidartinib) / Daiichi Sankyo           
          
            
             
dactolisib (RTB101) / Adicet Bio           
          
            
             
Cosela (trilaciclib) / G1 Therap           
          
            
             
Krazati (adagrasib) / BMS           
          
            
             
volasertib (NBL-001) / Oncoheroes, Notable Labs           
          
            
             
gedatolisib (PF-05212384) / Celcuity           
          
            
             
sotrastaurin (AEB071) / Novartis           
          
            
             
7-Hydroxystaurosporine (UCN-01) / National Cancer Institute           
          
            
             
afuresertib (LAE002) / Laekna Therap           
          
            
             
Fyarro (nanoparticle albumin-bound rapamycin) / Aadi Biosci           
          
            
             
avutometinib (VS-6766) / Verastem           
          
            
             
vactosertib (TEW-7197) / National OncoVenture, Theragen Etex           
          
            
            


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