Sarcoma  >>  c-KIT 


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 Phase 
N/A
1
2
3
4
 Trials
 021426384105126147168189210
            
            
             
imatinib / Generic mfg.           
          
            
             
sunitinib / Generic mfg.           
          
            
             
Votrient (pazopanib) / Novartis, BeiGene           
          
            
             
Focus V (anlotinib) / Advenchen, Sino Biopharm           
          
            
             
AiTan (rivoceranib) / HLB Bio Group           
          
            
             
sorafenib / Generic mfg.           
          
            
             
Stivarga (regorafenib) / Bayer           
          
            
             
Cabometyx (cabozantinib tablet) / Exelixis, Ipsen           
          
            
             
Tasigna (nilotinib) / Novartis, Inhibikase           
          
            
             
Ayvakit (avapritinib) / Blueprint Medicines           
          
            
             
Lenvima (lenvatinib) / Eisai, Merck (MSD)           
          
            
             
Qinlock (ripretinib) / Ono Pharma           
          
            
             
Cometriq (cabozantinib capsule) / Exelixis, Ipsen           
          
            
             
dasatinib / Generic mfg.           
          
            
             
famitinib (SHR 1020) / Jiangsu Hengrui Pharma           
          
            
             
Turalio (pexidartinib) / Daiichi Sankyo           
          
            
             
Kinaction (masitinib) / AB Science           
          
            
             
dovitinib (TKI258) / Novartis, Oncoheroes           
          
            
             
ganetespib (ADX-1612) / Aldeyra           
          
            
             
bezuclastinib (PLX9486) / Cogent Biosci           
          
            
             
motesanib (AMG 706) / Takeda           
          
            
             
vatalanib (PTK787) / Novartis, Bayer           
          
            
             
Balversa (erdafitinib) / J&J           
          
            
             
Fotivda (tivozanib) / Kyowa Kirin, Jazz, LG Chem           
          
            
             
Iclusig (ponatinib) / Takeda, Otsuka           
          
            
             
chiauranib (CS 2164) / Chipscreen           
          
            
             
tandutinib (MLN518) / Takeda           
          
            
             
Nailike (olverembatinib) / Ascentage Pharma, Takeda           
          
            
             
XL820 / Exelixis           
          
            
             
sitravatinib (MGCD516) / BeiGene