- |||||||||| Retrospective data, Review, Journal, Metastases: Efficacy of ALK inhibitors in Asian patients with ALK inhibitor-na (Pubmed Central) - Sep 12, 2024
Eight studies, involving 1,477 Asian patients and seven treatments (crizotinib, alectinib, brigatinib, ensartinib, envonalkib, iruplinalkib, and lorlatinib), were included in the NMA. Next-generation ALK inhibitors had better efficacy than crizotinib in the treatment of Asian patients with ALK inhibitor-na
- |||||||||| conteltinib (SY-707) / Centaurus Biopharma, Shouyao Holdings, SY-5933 / Shouyao Holdings
Targeting FAK to improve the therapy of KRAS G12C mutant cancers (Section 24) - Mar 5, 2024 - Abstract #AACR2024AACR_4014; In conclusion, our results demonstrate that CT-707 has the potential to enhance the efficacy of SY-5933 by suppressing adaptive FAK activation under KRAS G12C inhibition. This provides a rationale for an innovative combination therapy to improve outcomes in patients with KRAS G12C mutated cancers.
- |||||||||| Review, Journal: Roles and inhibitors of FAK in cancer: current advances and future directions. (Pubmed Central) - Feb 27, 2024
This review aims to clarify FAK's role in cancer, offering a comprehensive overview of the current status and future prospects of FAK-targeted therapy and combination approaches. The goal is to provide valuable insights for advancing anti-cancer treatment strategies.
- |||||||||| ficonalkib (SY-3505) / Shouyao Holdings
Trial completion date, Trial initiation date, Trial primary completion date, Metastases: A Study of SY-3505 in Patients With Advanced LTK Fusion-Positive Solid Tumors (clinicaltrials.gov) - Feb 15, 2024 P1, N=38, Recruiting, The goal is to provide valuable insights for advancing anti-cancer treatment strategies. Trial completion date: Dec 2025 --> May 2026 | Initiation date: Oct 2023 --> May 2024 | Trial primary completion date: Jun 2025 --> Dec 2025
- |||||||||| SY-4835 / Shouyao Holdings
Trial completion date, Trial primary completion date, Metastases: A Phase I Study of SY-4835 in Patients With Advanced Solid Tumors (clinicaltrials.gov) - Feb 15, 2024 P1, N=40, Recruiting, Trial completion date: Dec 2025 --> May 2026 | Initiation date: Oct 2023 --> May 2024 | Trial primary completion date: Jun 2025 --> Dec 2025 Trial completion date: Dec 2023 --> Dec 2024 | Trial primary completion date: Nov 2023 --> Jun 2024
- |||||||||| SY-4798 / Shouyao Holdings
Trial completion date, Trial primary completion date, Metastases: A First-in-Human, Phase 1 Study of SY-4798 in Patients With Advanced Solid Tumor (clinicaltrials.gov) - May 11, 2023 P1, N=80, Recruiting, Trial completion date: Dec 2023 --> Dec 2024 | Trial primary completion date: Nov 2023 --> Jun 2024 Trial completion date: Apr 2023 --> Apr 2024 | Trial primary completion date: Apr 2023 --> Apr 2024
- |||||||||| SY-4835 / Shouyao Holdings
Trial completion date, Trial primary completion date, Metastases: A Phase I Study of SY-4835 in Patients With Advanced Solid Tumors (clinicaltrials.gov) - Apr 12, 2023 P1, N=40, Recruiting, Trial primary completion date: Mar 2023 --> Jan 2025 Trial completion date: Jul 2023 --> Dec 2023 | Trial primary completion date: Jun 2023 --> Nov 2023
- |||||||||| ficonalkib (SY-3505) / Shouyao Holdings
Phase classification, Enrollment change, Trial completion date, Trial primary completion date, Metastases: Phase I/II Study of SY-3505 in Patients With ALK-positive Advanced Non-small Cell Lung Cancer (clinicaltrials.gov) - Feb 14, 2023 P1/2, N=150, Recruiting, Phase classification: P1 --> P1/2 | N=80 --> 200 | Trial completion date: Jun 2023 --> Feb 2025 Phase classification: P1 --> P1/2 | N=70 --> 150 | Trial completion date: Dec 2022 --> Aug 2024 | Trial primary completion date: Nov 2022 --> Apr 2024
- |||||||||| conteltinib (SY-707) / Centaurus Biopharma, Shouyao Holdings, Loqtorzi (toripalimab-tpzi) / Shanghai Junshi Biosci, Coherus Biosci
New P1/2 trial, Combination therapy, Metastases: Safety, Pharmacokinetics and Efficacy of CT-707, Toripalimab and Gemcitabine in Advanced Pancreatic Cancer (clinicaltrials.gov) - Oct 14, 2022 P1/2, N=114, Recruiting,
- |||||||||| conteltinib (CT-707) / Centaurus Biopharma, Nexavar (sorafenib) / Bayer, Amgen
Journal: CT-707 overcomes hypoxia-mediated sorafenib resistance in Hepatocellular carcinoma by inhibiting YAP signaling. (Pubmed Central) - Apr 27, 2022 TQ-B3139 was well-tolerated and exhibited promising anti-tumor activities in patients with ALK and ROS1 positive advanced NSCLC. Overall, this study not only favors the development of this novel multi-kinase inhibitor CT-707 as a therapeutic agent against HCC, but also provides a potential strategy to overcome the hypoxia-mediated resistance to sorafenib in HCC patients.
- |||||||||| SY-5007 / Shouyao Holdings
Trial primary completion date, Metastases: Phase I/II Study of SY-5007, a RET Inhibitor, in Patients With RET-altered Advanced Solid Tumor (clinicaltrials.gov) - Apr 7, 2022 P1, N=80, Recruiting, Overall, this study not only favors the development of this novel multi-kinase inhibitor CT-707 as a therapeutic agent against HCC, but also provides a potential strategy to overcome the hypoxia-mediated resistance to sorafenib in HCC patients. Trial primary completion date: Mar 2022 --> Mar 2023
- |||||||||| Anluoqing (envonalkib) / Sino Biopharm, Shouyao Holdings
Enrollment open, Trial primary completion date: Effect of High-fat Meal on the Pharmacokinetics of TQ-B3139 Capsules (clinicaltrials.gov) - Apr 1, 2021 P1, N=12, Recruiting, The dose-expansion phase of this study is ongoing. Not yet recruiting --> Recruiting | Trial primary completion date: Mar 2021 --> Mar 2022
- |||||||||| Anluoqing (envonalkib) / Sino Biopharm, Shouyao Holdings
Enrollment open, Trial initiation date, Metastases: A Phase I Study of TQ-B3139 on Tolerance and Pharmacokinetics (clinicaltrials.gov) - Sep 18, 2017 P1, N=20, Recruiting, Not yet recruiting --> Recruiting Not yet recruiting --> Recruiting | Initiation date: Mar 2017 --> Jul 2017
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