- |||||||||| grapiprant (RQ-00000007) / AskAt, Ikena Oncology, Maruishi Pharma
Enrollment closed, Combination therapy, PD(L)-1 Biomarker, Metastases: KEYNOTE-878: Grapiprant and Pembrolizumab in Patients With Advanced or Progressive MSS Colorectal Cancer (clinicaltrials.gov) - May 29, 2019 P1b, N=25, Active, not recruiting, Recruiting --> Active, not recruiting
- |||||||||| Journal: Aberrant FGFR signaling mediates resistance to CDK4/6 inhibitors in ER+ breast cancer. (Pubmed Central) - Apr 23, 2019
Addition of the FGFR TKI erdafitinib to palbociclib/fulvestrant induced complete responses of FGFR1-amplified/ER+ patient-derived-xenografts...Finally, ctDNA from patients enrolled in MONALEESA-2, the registration trial of ribociclib, showed that patients with FGFR1 amplification exhibited a shorter progression-free survival compared to patients with wild type FGFR1. Thus, we propose breast cancers with FGFR pathway alterations should be considered for trials using combinations of ER, CDK4/6 and FGFR antagonists.
- |||||||||| grapiprant (RQ-00000007) / AskAt, Ikena Oncology, Maruishi Pharma
Enrollment open, Combination therapy, PD(L)-1 Biomarker, Metastases: KEYNOTE-888: Grapiprant (ARY-007) and Pembrolizumab in Patients With Advanced or Metastatic Post-PD-1/L1 NSCLC Adenocarcinoma (clinicaltrials.gov) - Dec 20, 2018 P1b/2, N=25, Recruiting, Thus, we propose breast cancers with FGFR pathway alterations should be considered for trials using combinations of ER, CDK4/6 and FGFR antagonists. Not yet recruiting --> Recruiting
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Trial termination, Metastases: A Study to Assess the Efficacy and Safety of the VEGFR-FGFR Inhibitor, Lucitanib, Given to Patients With Advanced/Metastatic Lung Cancer and FGF, VEGF, or PDGF Related Genetic Alterations (clinicaltrials.gov) - Sep 18, 2018 P2, N=18, Terminated, Not yet recruiting --> Recruiting Completed --> Terminated
- |||||||||| Liporaxel (paclitaxel oral) / Dae Hwa, HaiHe Biopharma
Enrollment open, Trial completion date, Trial initiation date, Trial primary completion date, Metastases: OPERA: Oral Paclitaxel Efficacy Safety and PK in Recurrent and Metastatic Breast Cancer (clinicaltrials.gov) - Aug 13, 2018 P2, N=72, Recruiting, Active, not recruiting --> Completed Not yet recruiting --> Recruiting | Trial completion date: Jan 2019 --> Sep 2019 | Initiation date: Dec 2017 --> Jul 2018 | Trial primary completion date: Sep 2018 --> May 2019
- |||||||||| Liporaxel (paclitaxel oral) / Dae Hwa, HaiHe Biopharma
Enrollment open, Trial completion date, Trial primary completion date, Metastases: OPTIMAL: Oral Paclitaxel Trial In Recurrent and Metastatic Breast Cancer As 1st Line Therapy (clinicaltrials.gov) - Jun 6, 2018 P2/3, N=476, Recruiting, Not yet recruiting --> Recruiting | Trial completion date: Jan 2019 --> Sep 2019 | Initiation date: Dec 2017 --> Jul 2018 | Trial primary completion date: Sep 2018 --> May 2019 Not yet recruiting --> Recruiting | Trial completion date: Oct 2021 --> Mar 2022 | Trial primary completion date: Oct 2018 --> Jan 2019
- |||||||||| delpazolid (LCB01-0371) / LegoChem Biosci
Trial completion date, Trial primary completion date: A Phase II Clinical Study of LCB01-0371 to Evaluate the EBA, Safety and PK (clinicaltrials.gov) - Apr 10, 2018 P2, N=64, Recruiting, Therefore, these tumors are endocrine resistant and should be candidates for treatment with combinations of ER and FGFR antagonists. Trial completion date: Feb 2018 --> Dec 2018 | Trial primary completion date: Feb 2018 --> Oct 2018
- |||||||||| delpazolid (LCB01-0371) / LegoChem Biosci
Trial completion, Trial completion date: IV Dosage Form of LCB01-0371 Phase I Study in Healthy Male Volunteers (clinicaltrials.gov) - Apr 10, 2018 P1, N=24, Completed, Trial completion date: Feb 2018 --> Dec 2018 | Trial primary completion date: Feb 2018 --> Oct 2018 Recruiting --> Completed | Trial completion date: Dec 2017 --> Jul 2017
- |||||||||| delpazolid (LCB01-0371) / LegoChem Biosci
Enrollment open, Enrollment change, Trial primary completion date: A Phase II Clinical Study of LCB01-0371 to Evaluate the EBA, Safety and PK (clinicaltrials.gov) - Aug 29, 2017 P2, N=64, Recruiting, Phase classification: P1a/1b --> P1 Not yet recruiting --> Recruiting | N=30 --> 64 | Trial primary completion date: May 2017 --> Feb 2018
- |||||||||| simmitecan / HaiHe Biopharma, Shanghai Inst. of Materia Medica
Enrollment change, Trial primary completion date, Monotherapy, Metastases: Study to Evaluate the Safety, Tolerability, Preliminary Efficacy and Pharmacokinetics of Simmitecan Monotherapy and Combination in Patients With Advanced Solid Tumors (clinicaltrials.gov) - Jul 17, 2017 P1, N=243, Recruiting, Not yet recruiting --> Recruiting | N=30 --> 64 | Trial primary completion date: May 2017 --> Feb 2018 N=158 --> 243 | Trial primary completion date: Oct 2018 --> Dec 2020
- |||||||||| grapiprant (RQ-00000007) / AskAt, Ikena Oncology, Maruishi Pharma
Enrollment change, Trial initiation date, Trial withdrawal, Metastases: Phase II Trial of EP4 Receptor Antagonist, AAT-007 (RQ-07; CJ-023,423) in Advanced Solid Tumors (clinicaltrials.gov) - Jun 7, 2017 P2, N=0, Withdrawn, N=158 --> 243 | Trial primary completion date: Oct 2018 --> Dec 2020 N=45 --> 0 | Initiation date: Jan 2017 --> Jun 2017 | Not yet recruiting --> Withdrawn
- |||||||||| simmitecan / HaiHe Biopharma, Shanghai Inst. of Materia Medica
Enrollment open, Monotherapy, Metastases: Study to Evaluate the Safety, Tolerability, Preliminary Efficacy and Pharmacokinetics of Simmitecan Monotherapy and Combination in Patients With Advanced Solid Tumors (clinicaltrials.gov) - Mar 22, 2017 P1, N=158, Recruiting, Active, not recruiting --> Completed | N=123 --> 76 Not yet recruiting --> Recruiting
- |||||||||| delpazolid (LCB01-0371) / LegoChem Biosci
Enrollment open, Trial primary completion date: IV Dosage Form of LCB01-0371 Phase I Study in Healthy Male Volunteers (clinicaltrials.gov) - Mar 13, 2017 P1, N=24, Recruiting, Not yet recruiting --> Recruiting Not yet recruiting --> Recruiting | Trial primary completion date: Dec 2016 --> Sep 2017
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Trial completion, Trial primary completion date, Metastases: A Study to Assess the Efficacy and Safety of the VEGFR-FGFR Inhibitor, Lucitanib, Given to Patients With Advanced/Metastatic Lung Cancer and FGF, VEGF, or PDGF Related Genetic Alterations (clinicaltrials.gov) - Nov 14, 2016 P2, N=18, Completed, Active, not recruiting --> Completed Active, not recruiting --> Completed | Trial primary completion date: Sep 2016 --> Apr 2016
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Enrollment change, Trial initiation date, Trial withdrawal, Trial primary completion date, Pan tumor, Metastases: Lucitanib (E3810) in Patients With Advanced Cancer and FGFR, VEGFR, or PDGFR Pathway Aberrations (clinicaltrials.gov) - Nov 2, 2016 P2, N=0, Withdrawn, Active, not recruiting --> Completed | Trial primary completion date: Sep 2016 --> Apr 2016 N=180 --> 0 | Initiation date: Apr 2016 --> Apr 2017 | Not yet recruiting --> Withdrawn | Trial primary completion date: Apr 2020 --> Apr 2021
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Trial primary completion date, Metastases: A Study to Assess the Efficacy and Safety of the VEGFR-FGFR Inhibitor, Lucitanib, Given to Patients With Advanced/Metastatic Lung Cancer and FGF, VEGF, or PDGF Related Genetic Alterations (clinicaltrials.gov) - Jul 28, 2016 P2, N=18, Active, not recruiting, Recruiting --> Active, not recruiting Trial primary completion date: Jun 2016 --> Sep 2016
- |||||||||| grapiprant (RQ-00000007) / AskAt, Ikena Oncology, Maruishi Pharma
Trial initiation date, Trial primary completion date, Metastases: Phase II Trial of EP4 Receptor Antagonist, AAT-007 (RQ-07; CJ-023,423) in Advanced Solid Tumors (clinicaltrials.gov) - May 23, 2016 P2, N=45, Not yet recruiting, Trial primary completion date: Jun 2016 --> Sep 2016 Initiation date: Dec 2015 --> Jan 2017 | Trial primary completion date: Dec 2017 --> Dec 2019
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Enrollment closed, Metastases: A Study to Assess the Safety and Efficacy of the VEGFR-FGFR-PDGFR Inhibitor, Lucitanib, Given to Patients With Metastatic Breast Cancer (clinicaltrials.gov) - Apr 7, 2016 P2, N=178, Active, not recruiting, Recruiting --> Terminated Recruiting --> Active, not recruiting
- |||||||||| simmitecan / HaiHe Biopharma
Enrollment closed, Enrollment change, Trial primary completion date, Metastases: Study of Simmitecan Hydrochloride in the Treatment of Advanced Solid Tumor (clinicaltrials.gov) - Mar 21, 2016 P1, N=39, Active, not recruiting, Not yet recruiting --> Completed | N=24 --> 30 | Trial primary completion date: Sep 2015 --> Dec 2015 Recruiting --> Active, not recruiting | N=51 --> 39 | Trial primary completion date: Jan 2014 --> Mar 2016
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Trial primary completion date, Metastases: Study of Oral Lucitanib (E-3810), a Dual VEGFR-FGFR Tyrosine Kinase Inhibitor, in Patients With Solid Tumors (clinicaltrials.gov) - Mar 14, 2016 P1/2, N=130, Active, not recruiting, Recruiting --> Active, not recruiting | N=51 --> 39 | Trial primary completion date: Jan 2014 --> Mar 2016 Trial primary completion date: Dec 2015 --> Sep 2016
- |||||||||| lucitanib (E 3810) / Clovis, Servier
Enrollment closed, Enrollment change, Metastases: A Study to Assess the Efficacy and Safety of the VEGFR-FGFR Inhibitor, Lucitanib, Given to Patients With Advanced/Metastatic Lung Cancer and FGF, VEGF, or PDGF Related Genetic Alterations (clinicaltrials.gov) - Jan 21, 2016 P2, N=18, Active, not recruiting, Trial primary completion date: Dec 2015 --> Sep 2016 Recruiting --> Active, not recruiting | N=40 --> 18
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