- |||||||||| Zepzelca (lurbinectedin) / PharmaMar, Jazz, Tecentriq (atezolizumab) / Roche
New P1 trial, PD(L)-1 Biomarker, Metastases: 2SMALL: Study to Assess Safety,Tolerability,Efficacy of PM01183 and Atezolizumab in Patients w/ Advanced Small Cell Lung Cancer. (clinicaltrials.gov) - Feb 4, 2020 P1, N=25, Recruiting,
- |||||||||| Yondelis (trabectedin) / Otsuka, PharmaMar, Valeo Pharma, Zepsyre (lurbinectedin) / PharmaMar, Jazz
Journal: The antitumor drugs trabectedin and lurbinectedin induce transcription-dependent replication stress and genome instability. (Pubmed Central) - Jan 27, 2020 Given the increasing evidence that R-loops occur all over the genome, the ability of lurbinectedin and trabectedin to act on them may contribute to enhance their efficacy, opening the possibility that R-loops might be a feature shared by specific cancers. Implications: The data presented in this study provide the new concept that R-loops are important cellular factors that contribute to trabectedin and lurbinectedin anticancer activity.
- |||||||||| fimasartan (BR-A-657) / Boryung Group
Clinical, Journal: Fimasartan reduces clinic and home pulse pressure in elderly hypertensive patients: A K-MetS study. (Pubmed Central) - Dec 23, 2019 Implications: The data presented in this study provide the new concept that R-loops are important cellular factors that contribute to trabectedin and lurbinectedin anticancer activity. Fimasartan resulted in better pulse pressure reduction with similar BP reduction efficacy and safety in hypertensive elderly patients compared with nonelderly patients.
- |||||||||| Zepzelca (lurbinectedin) / PharmaMar, Jazz
Phase classification, Enrollment change, Trial completion date, Trial primary completion date, Combination therapy, Metastases: PM1183-A-014-15: Pharmacokinetic Study of Lurbinectedin in Combination With Irinotecan in Patients With Selected Solid Tumors (clinicaltrials.gov) - Dec 23, 2019 P1/2, N=150, Recruiting, In a word, this study may provide more information for understanding the effect of inhibition of the aplidin on the LMW-PTP. Phase classification: P1 --> P1/2 | N=100 --> 150 | Trial completion date: May 2020 --> Nov 2021 | Trial primary completion date: May 2019 --> Nov 2020
- |||||||||| fimasartan (BR-A-657) / Boryung Group
Retrospective data, Review, Journal, Combination therapy: Systematic Review with Network Meta-Analysis: Comparative Efficacy and Safety of Combination Therapy with Angiotensin II Receptor Blockers and Amlodipine in Asian Hypertensive Patients. (Pubmed Central) - Dec 14, 2019 The analysis included 1198 Asian HTN patients from seven studies involving six ARB-AML CTs: azilsartan (AZL), candesartan (CAN), fimasartan (FIM), losartan (LOS), olmesartan (OLM), and telmisartan (TEL)...Safety profiles among the ARB-AML CTs were largely comparable. Due to the limited study size and small number of trials (direct evidence), our findings should best be interpreted as an exploratory effort importance to inform future research direction.
- |||||||||| Kanarb (fimasartan) - Boryung Group, R / Pharm
Trial completion, Trial completion date: FABULOUS: Fimasartan Blood Pressure Lowering After Acute Stroke (clinicaltrials.gov) - Nov 4, 2019 P=N/A, N=1035, Completed, Active, not recruiting --> Completed Recruiting --> Completed | Trial completion date: Dec 2019 --> Apr 2019
- |||||||||| Clinical, Review, Journal: Marine-Derived Anticancer Agents: Clinical Benefits, Innovative Mechanisms, and New Targets. (Pubmed Central) - Nov 2, 2019
Approximately 50 years since the approval of cytarabine, the marine-derived anticancer pharmaceutical pipeline includes four approved drugs and eighteen agents in clinical trials, six of which are in late development. Thus, the dynamic pharmaceutical pipeline consisting of approved and developmental marine-derived anticancer agents offers new hopes and new tools in the treatment of patients afflicted with previously intractable types of cancer.
- |||||||||| Zepsyre (lurbinectedin) / PharmaMar
Journal, Checkpoint inhibition: Lurbinectedin synergizes with immune checkpoint blockade to generate anticancer immunity. (Pubmed Central) - Oct 26, 2019 Anticancer effects resulting from lurbinectedin treatment were boosted in combination with PD-1 and CTLA-4 double immune checkpoint blockade (ICB), and lurbinectedin combined with double ICB exhibited strong antineoplastic effects. Cured animals exhibited long term immune memory effects that rendered them resistant to rechallenge with syngeneic tumors underlining the potency of combination therapy with lurbinectedin.
- |||||||||| Zepsyre (lurbinectedin) / PharmaMar
Lurbinectedin down-regulates ASCL1 transcription factor in Small Cell Lung Cancer (SCLC) (Board 161: Level 2 - Hall D) - Oct 25, 2019 - Abstract #AACRNCIEORTC2019AACR_NCI_EORTC_684; We tested whether lurbinectedin shared a similar effect on transcriptomic profile as other known drug by dividing up and down regulated genes and testing their correlation to the drug-related gene profiles provided by the tool Enrichr, we found that lurbinectedin has a high correlation to the topoisomerase I inhibitor class. This finding deserves further experimental verifications also in view of potential clinical interest in the combination of lurbinectedin and topoisomerase I inhibitors.
- |||||||||| Aplidin (plitidepsin) / PharmaMar, Roche
Review, Journal: Plitidepsin for multiple myeloma. (Pubmed Central) - Oct 22, 2019 This finding deserves further experimental verifications also in view of potential clinical interest in the combination of lurbinectedin and topoisomerase I inhibitors. No abstract available
- |||||||||| paclitaxel / Generic Mfg.
Subungual metastasis of an endometrial carcinoma () - Oct 16, 2019 - Abstract #ESGO2019ESGO_1231; A weekly Carboplatinum and Paclitaxel chemotherapy with concomitant Denosumab was initiated...As confirmed by the literature, the occurrence of subungual metastasis is precursor to the rapid fatal progression of the disease. Beside the unexpected topography of the metastasis, the absence of an underlying bone involvement and the mild clinical manifestations were singular features of this progression pattern.
- |||||||||| Kanarb (fimasartan) - Boryung Group, R / Pharm
Enrollment closed, Trial completion date, Trial primary completion date: A Randomized, Double-blind, Active Control, Parallel Group, Titration, Multicenter Study to Evaluate the Efficacy and Safety of Fimasartan (clinicaltrials.gov) - Sep 18, 2019 P3, N=468, Active, not recruiting, Oral administration of F/A 10 mg/kg could improve LV systolic function and reduce infarct size in a rat MI model. Recruiting --> Active, not recruiting | Trial completion date: Dec 2020 --> Jun 2022 | Trial primary completion date: Dec 2018 --> Dec 2019
- |||||||||| fimasartan (BR-A-657) / Boryung Group
Review, Journal: Fimasartan: A new armament to fight hypertension. (Pubmed Central) - Aug 30, 2019 Further, it is renoprotective and has proven beneficial in diabetes also. This article briefly discusses the pharmacology and clinical evidence with fimasartan with a short summary of previous angiotensin receptor blockers.
- |||||||||| Aplidin (plitidepsin) / PharmaMar, Roche
Clinical, P3 data, Clinical Trial,Phase I, Clinical Trial,Phase II, Clinical Trial,Phase III, Journal, Combination therapy: Randomized phase III study (ADMYRE) of plitidepsin in combination with dexamethasone vs. dexamethasone alone in patients with relapsed/refractory multiple myeloma. (Pubmed Central) - Aug 29, 2019 The safety profile does not overlap with the toxicity observed with other agents used in multiple myeloma. In conclusion, efficacy data, the reassuring safety profile, and the novel mechanism of action of plitidepsin suggest that this combination can be an alternative option in patients with relapsed/refractory multiple myeloma after at least three prior therapy lines.
- |||||||||| Zepsyre (lurbinectedin) / PharmaMar
Journal, BRCA Biomarker: Lurbinectedin for BRCA-mutated advanced breast cancer. (Pubmed Central) - Jun 15, 2019 Similar, main pharmacokinetic parameters were calculated with the concentrations obtained either thru this method or by using a chemically synthetized authentic standard. No abstract available
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